A selective c-Met inhibitor (IC50 = 3 nM) that inhibits c-Met phosphorylation and downstream signaling in various cancer cell lines (IC50s = 6-9 nM) and at 5-15 mg/kg regresses tumors in mouse xenograft models
产品描述
A selective c-Met inhibitor (IC50 = 3 nM) that inhibits c-Met phosphorylation and downstream signaling in various cancer cell lines (IC50s = 6-9 nM) and at 5-15 mg/kg regresses tumors in mouse xenograft models