(R,S)-Atenolol is a β1-adrenergic receptor antagonist with Ki values of 1.14 and 48.7 µM for β1 and β2, respectively.{28226} It has been reported that only the (S) enantiomer contributes to the beta-blocking effects of racemic atenolol.{28227,25396} Beta-blockers, including atenolol, have diverse applications in cardiology and vascular disease.{25151}
产品描述
A β1-adrenergic receptor antagonist (Kis = 1.14 and 48.7 µM for β1 and β2, respectively); has applications in cardiology and vascular disease